ENDOTHELIN ANTAGONISTS: N-[[2'-[[(4,5-DIMETHYL-3-ISOXAZOLYL) AMINO] SULFONYL]-4-(2-OXAZOLYL) [1,1'-BIPHENYL]-2-YL] METHYL]-N-3,3-TRIMETHYLBUTANAMIDE) AND SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM
申请(专利)号:
IL19980130622
申请日期:
1998-01-26
公开/公告号:
IL130622A
公开/公告日期:
2003-01-12
申请(专利权)人:
BRISTOL-MYERS SQUIBB COMPANY
摘要:
The compounds N-[[2'-[[(4,5-dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]-2-yl]methyl]-N,3,3-trimethylbutanamide and N-(4,5-dimethyl-3-isoxazolyl)-2'-[(3,3-dimethyl-2-oxo-1-pyrrolidinyl)methyl]-4'-(2-oxazolyl)[1,1'-biphenyl]-2-sulfonamide, and salts thereof, useful as endothelin antagonists.
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