ENDOTHELIN ANTAGONISTS: N-[[2'-[[(4,5-DIMETHYL-3-ISOXAZOLYL) AMINO] SULFONYL]-4-(2-OXAZOLYL) [1,1'-BIPHENYL]-2-YL] METHYL]-N-3,3-TRIMETHYLBUTANAMIDE) AND SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM

阅读量:

5

申请(专利)号:

IL19980130622

申请日期:

1998-01-26

公开/公告号:

IL130622A

公开/公告日期:

2003-01-12

申请(专利权)人:

BRISTOL-MYERS SQUIBB COMPANY

摘要:

The compounds N-[[2'-[[(4,5-dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]-2-yl]methyl]-N,3,3-trimethylbutanamide and N-(4,5-dimethyl-3-isoxazolyl)-2'-[(3,3-dimethyl-2-oxo-1-pyrrolidinyl)methyl]-4'-(2-oxazolyl)[1,1'-biphenyl]-2-sulfonamide, and salts thereof, useful as endothelin antagonists.

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