摘要：

A number of phenolic compounds were readily aminoalkylated at room temperature by reaction with dihydro-2H-1,3-benzoxazines to give high yields of tertiary amines having two hydroxybenzyl groups attached to nitrogen. This novel aminoalkylation reaction occurred preferentially at the ortho position of phenols containing both free ortho and para positions. Major differences were observed in the behavior of benzoxazines and analogous naphthoxazines in the reaction.

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