Efficient and simple synthesis of 3-aryl-1H-pyrazoles - ScienceDirect

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作者：

Anne-Laure，Gérard，and，Alexandre，Bouillon，and，Clément，Mahatsekake，and，Valérie

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摘要：

Efficient preparation of 3-aryl-1H-pyrazoles by reaction of 1-protected-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazoles with (het)aryl halides is described. The choice of THP protecting group is discussed.

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关键词：

pyrazole derivatives protection, deprotection C‐C bond formation

DOI：

10.1016/j.tetlet.2006.04.125

被引量：

190

年份：

2006

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来源期刊

Tetrahedron Letters

3 July 2006

引用走势

2009

被引量：43

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