Pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present

The present invention relates to compounds of the formula: ##STR1## These compounds are useful in pharmaceuticals in which cannabis is known to be involved.

F Barth，P Casellas，C Congy，... - US

Antihypercholesterolemic compounds

6(R)- 2-(8'-acyloxy-2'-methyl-6'-methyl (or hydrogen)- polyhydronaphthyl-1')-ethyl!-4(R)-hydroxy-3,4,5,6-tetrahydro-2H-p yran-2- ones are prepared by acylation of the corresponding 8'-hydroxy compounds. The products are strong inhibitor...

WF Hoffman，RL Smith，AK Willard - US

Antihypercholesterolemic compounds

6(R)- 2-(8'-acyloxy-2'-methyl-6'-methyl (or hydrogen)- polyhydronaphthyl-1')-ethyl!-4(R)-hydroxy-3,4,5,6-tetrahydro-2H-p yran-2- ones are prepared by acylation of the corresponding 8'-hydroxy compounds. The products are strong inhibitor...

 - US

N-substituted pseudo-aminosugars, their production and use

These compounds exhibit excellent inhibitory activity against α-glucoside hydrolase, thus are useful for hyperglycemic symptoms and various disorders caused by hyperglycemia.

H Fukase，S Horii，Y Kameda - US

Bicarbocyclic aryl urea or thiourea compounds

The invention relates primarily to pharmaceutical compositions and medicaments containing a compound of Formula (I), infra as the active ingredient. Also i...

HJ Kabbe，E Klauke，HP Krause，... - US

Pharmaceutically acceptable salts

Improved pharmaceutical salts of amlodipine, particularly the besylate salt, and pharmaceutical compositions thereof. These salts find utility as anti-ischaemic and anti-hypertensive agents.

E Davison，JI Wells - US

Biomass lipase inhibitor useful for treating adiposity

A pharmaceutical composition comprising at least one water insoluble crude fiber and at least one lipase inhibitor. The lipase inhibitor is present in an amount effective for treating adiposity. The lipase inhibitor is selected from lips...

D Isler，W Rehm，E Widmer - US

Cholesteryl ester transfer protein inhibitors which are used to elevate highdensity lipoprotein-cholesterol and to lower low density lipoprotein-cholestero...

Cholesteryl ester transfer protein inhibitors, pharmaceutical compositions containing such inhibitors and the use of such inhibitors to elevate certain pla...

MP Deninno，GT Magnus-Aryitey，RB Ruggeri，... - US

Physiologically active substances

Physiologically active substances ML-236 of the formula ##SPC1## Wherein R is hydrogen atom, hydroxy group or 2-methylbutyryloxy group having cholesterol- and lipid-lowering effects in blood and liver and thus utility as hypocholesteremi...

A Endo，M Kuroda，A Terahara，... - US

Anticholesterol agents

Cholesteryl ester transfer protein inhibitors, pharmaceutical compositions containing such inhibitors and the use of such inhibitors to elevate certain pla...

MP Deninno，GT Magnus-Aryitey，RB Ruggeri，...