From a broad screening program, the 4-hydroxycoumarin phenprocoumon (I) was previously identified as a lead template with HIV protease inhibitory activity....
The corresponding derivatives of Δ 1,3,5(10),9,(11)-8,14-seco- d-homo-oestratetraen-3-ol-14,17a-dione(VII, VIII, IX) have been obtained by the condensation of 3-methoxy-, 3-hydroxy-, and 3-tetrahydropyranyloxy-1-vinyltetralols (IV, V, V...
Larvicidal activity against the beet armyworm, Spodoptera exigua (H眉bner), was measured after topical treatment for a series of N-tert-butyl-dibenzoylhydr...
To develop antagonists which show selectivity in blocking neurotransmitters, several aminophosphonoic acids, 2-amino-5-phosphonopentanoic acid (IVb), 2-ami...
To develop antagonists which show selectivity in blocking neurotransmitters, several aminophosphonoic acids, 2-amino-5-phosphonopentanoic acid (IVb), 2-ami...
Structural analogues and homologues of the raspberry ketone, 4-(p-hydroxyphenyl)-2-butanone, have been prepared. A systematic study of their organoleptic properties reveals that the structure of 4-(p-hydroxyphenyl)-2-butanone is highly s...
Some 6-arylthio( aryloxy and alkylthio )-3-( acetamidomethyl , benzamidomethyl, methoxy and unsubstituted )-2-arylimidazo[1,2-b] pyridazines have been prepared and examined for their ability to displace [3H]diazepam from rat brain membra...
Syntheses of DL-2-piperidinemethanol (XXXIII) and meso-cis-2, 6-piperidinedimethanol (XXXIV) were accomplished through a few steps from 2-picoline (I) and ...
Photomagnetic effects were recently evidenced in CoFe Prussian-blue analogues. In order to understand the mechanism and the scope of the phenomenon, we und...